SCHEMBL29449658

SCHEMBL29449658

COc1cc2ncnc(Nc3ccc([C@@H](C)NC(C)=O)cc3)c2cc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.58
RET P07949 5/20 0.58
KIF5B P33176 4/20 0.58
EGFR P00533 9/20 0.57
AURKB Q96GD4 2/20 0.57
RIPK2 O43353 2/20 0.57
JAK3 P52333 2/20 0.57
GAK O14976 1/20 0.57
STK10 O94804 1/20 0.57
FLT3 P36888 1/20 0.57
AAK1 Q2M2I8 1/20 0.57
Q6ZSR9 Q6ZSR9 1/20 0.57
SLK Q9H2G2 1/20 0.57
IRAK4 Q9NWZ3 1/20 0.57
RPS6KA6 Q9UK32 1/20 0.57
ALK Q9UM73 1/20 0.57
AURKA O14965 1/20 0.56
LCK P06239 3/20 0.56
ABCB1 P08183 1/20 0.53
ABCG2 Q9UNQ0 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29449673 1.00 KDR (0.58) KDRRETKIF5BEGFRAURKB
SCHEMBL28691068 1.00 KDR (0.58) KDRRETKIF5BEGFRAURKB
Hydrochloric Acid SCHEMBL28302017 0.99 EGFR (0.58) KDRRETKIF5BEGFRAURKB
SCHEMBL28694471 0.88 KDR (0.60) KDRRETEGFRAURKBRIPK2
SCHEMBL29449696 0.88 KDR (0.60) KDRRETEGFRAURKBRIPK2
SCHEMBL29449683 0.88 KDR (0.60) KDRRETEGFRAURKBRIPK2
SCHEMBL28985109 0.85 KDR (0.53) KDRRETKIF5BEGFRAURKB
SCHEMBL29449684 0.85 KDR (0.55) KDRRETKIF5BEGFRAURKB
SCHEMBL29449681 0.85 KDR (0.55) KDRRETKIF5BEGFRAURKB
SCHEMBL28689947 0.85 KDR (0.55) KDRRETKIF5BEGFRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942499-B Quinazoline derivative and preparation method and application thereof 湖南中医药大学 2022-03-22 CN disclosed