SCHEMBL29458570

SCHEMBL29458570

CC(F)CNCc1ccc(-c2nnc(-c3nc(-c4ccc(S(=O)(=O)C(C)CCO)cc4)cnc3N)o2)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.55
PRKDC P78527 4/20 0.48
GSK3B P49841 1/20 0.48
ATM Q13315 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3055564 1.00 ATR (0.55) ATRPRKDCGSK3BATM
SCHEMBL3059314 0.94 ATR (0.56) ATRPRKDCGSK3BATM
SCHEMBL3056584 0.92 ATR (0.57) ATRPRKDCGSK3BATM
SCHEMBL3056276 0.92 ATR (0.57) ATRPRKDCGSK3BATM
SCHEMBL29458691 0.91 ATR (0.49) ATRPRKDCGSK3B
SCHEMBL3059671 0.91 ATR (0.49) ATRPRKDCGSK3B
SCHEMBL16070059 0.91 ATR (0.55) ATRPRKDCGSK3BATM
SCHEMBL3042729 0.91 ATR (0.59) ATRPRKDCGSK3BATM
SCHEMBL29458664 0.91 ATR (0.59) ATRPRKDCGSK3BATM
SCHEMBL3048919 0.91 ATR (0.66) ATRPRKDCGSK3BATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3354650-B1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2022-02-16 EP disclosed