SCHEMBL29466293

SCHEMBL29466293

NC(=O)c1ccnc(Nc2ccccc2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 5/20 0.60
MAPK10 P53779 1/20 0.58
AURKA O14965 6/20 0.57
PRKCD Q05655 2/20 0.56
CHEK1 O14757 1/20 0.56
IKBKB O14920 1/20 0.56
NPC1 O15118 1/20 0.56
PDPK1 O15530 1/20 0.56
CHEK2 O96017 1/20 0.56
PRKCG P05129 1/20 0.56
CDK1 P06493 1/20 0.56
LYN P07948 1/20 0.56
MAPT P10636 1/20 0.56
KIT P10721 1/20 0.56
PIM1 P11309 1/20 0.56
FGFR1 P11362 1/20 0.56
FGFR3 P22607 1/20 0.56
RPS6KB1 P23443 1/20 0.56
CDK2 P24941 1/20 0.56
MARK3 P27448 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670431 0.87 KDM4E (0.62) MAPK8MAPK10AURKAPRKCDCHEK1
SCHEMBL29484634 0.87 AURKA (0.59) MAPK8MAPK10AURKAPRKCDCHEK1
SCHEMBL29938984 0.84 MAPT (0.58) MAPK8MAPK10AURKANPC1MAPT
SCHEMBL5598434 0.84 JAK2 (0.57) MAPK8MAPK10AURKAPRKCDCHEK1
SCHEMBL25882561 0.82 GSK3A (0.50) MAPK8AURKAPRKCDCHEK1IKBKB
SCHEMBL29466335 0.82 GSK3A (0.50) MAPK8AURKAPRKCDCHEK1IKBKB
SCHEMBL29466300 0.81 AURKA (0.45) MAPK8MAPK10AURKANPC1CDK1
SCHEMBL670174 0.81 AURKA (0.53) MAPK8AURKAPRKCDCHEK1IKBKB
SCHEMBL25883208 0.81 GSK3A (0.58) MAPK8AURKAPRKCDCHEK1IKBKB
SCHEMBL29939485 0.81 GSK3A (0.55) MAPK8MAPK10AURKAIKBKBKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110545817-B GSK-3 inhibitors 百时美施贵宝公司 2022-11-15 CN disclosed
CN-114195780-A Carbonyl heterocyclic compound and application thereof 上海医药集团股份有限公司 2022-03-18 CN disclosed
CN-114195806-A Carbonyl heterocyclic compound and application thereof 上海医药集团股份有限公司 2022-03-18 CN disclosed