SCHEMBL29482127

SCHEMBL29482127

CS(=O)(=O)N1CCN(Cc2cc3nc(-c4cccc5[nH]ccc45)nc(N4CCOCC4)c3s2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 18/20 1.00
PIK3CA P42336 16/20 0.80
PIK3CB P42338 15/20 0.80
PIK3CG P48736 15/20 0.80
PIK3C2A O00443 1/20 0.80
PLK4 O00444 1/20 0.80
PIK3R2 O00459 1/20 0.80
PIK3C2B O00750 1/20 0.80
GAK O14976 1/20 0.80
EPHB6 O15197 1/20 0.80
DAPK3 O43293 1/20 0.80
STK16 O75716 1/20 0.80
PIK3C2G O75747 1/20 0.80
NTRK1 P04629 1/20 0.80
NQO2 P16083 1/20 0.80
CSNK2A2 P19784 1/20 0.80
JAK1 P23458 1/20 0.80
PIK3R1 P27986 1/20 0.80
TYK2 P29597 1/20 0.80
AKT1 P31749 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL391747 1.00 PIK3CD (1.00) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A
SCHEMBL393696 0.90 PIK3CD (0.81) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2469939 0.90 PIK3CD (0.81) PIK3CDPIK3CAPIK3CBPIK3CG
Pictilisib SCHEMBL190812 0.89 PIK3CA (1.00) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A
Pictilisib SCHEMBL29387739 0.89 PIK3CA (1.00) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A
Pictilisib SCHEMBL14859338 0.89 PIK3CA (1.00) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A
Pictilisib SCHEMBL29375636 0.89 PIK3CA (1.00) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A
SCHEMBL2465953 0.89 PIK3CD (0.79) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2466623 0.89 PIK3CD (0.79) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL2436174 0.88 PIK3CA (0.80) PIK3CDPIK3CAPIK3CBPIK3CGPIK3C2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118994402-A Antibodies to PMEL17 and conjugates thereof 诺华股份有限公司 2024-11-22 CN disclosed
CN-113195541-B Antibodies to PMEL17 and conjugates thereof 诺华股份有限公司 2024-08-30 CN disclosed
CN-118420766-A Antibodies to PMEL17 and conjugates thereof 诺华股份有限公司 2024-08-02 CN disclosed
CN-110248963-B anti-CCR 7 antibody drug conjugates 诺华股份有限公司 2023-12-26 CN disclosed
CN-116096426-A CCR7 antibody drug conjugates for the treatment of cancer 诺华股份有限公司 2023-05-09 CN disclosed
CN-108341873-B Antibodies to epidermal growth factor receptor 3(HER3) 诺华股份有限公司 2022-03-25 CN disclosed