SCHEMBL29482190

SCHEMBL29482190

COC(=O)[C@@H](N)CCNC(=O)CCCCc1ccc2c(n1)NCCC2

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.68
ITGB3 P05106 18/20 0.68
ITGB6 P18564 10/20 0.58
ITGB5 P18084 9/20 0.56
ITGB8 P26012 8/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22029442 1.00 ITGAV (0.68) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL24193794 0.91 ITGAV (0.66) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL22029437 0.90 ITGAV (0.69) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL21706034 0.90 ITGAV (0.75) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL22029478 0.90 ITGAV (0.75) ITGAVITGB3ITGB6ITGB5ITGB8
SCHEMBL29813942 0.88 ITGAV (0.61) ITGAVITGB3ITGB6
SCHEMBL24683292 0.88 ITGAV (0.61) ITGAVITGB3ITGB6
SCHEMBL21852990 0.88 ITGAV (0.61) ITGAVITGB3ITGB6
SCHEMBL21852991 0.88 ITGAV (0.61) ITGAVITGB3ITGB6
SCHEMBL29813809 0.88 ITGAV (0.61) ITGAVITGB3ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3481814-B1 TETRAHYDRONAPHTHYRIDINEPENTANAMIDE INTEGRIN ANTAGONISTS UNIV ROCKEFELLER (US) 2022-04-27 EP disclosed