SCHEMBL29500488

SCHEMBL29500488

[2H]n1c(C2CC2)nc2cc(N)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
MAPT P10636 5/20 0.49
GFER P55789 3/20 0.49
RAB9A P51151 4/20 0.37
ALDH1A1 P00352 4/20 0.37
NPC1 O15118 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
HTT P42858 2/20 0.36
F2 P00734 1/20 0.36
LMNA P02545 1/20 0.36
CHRM2 P08172 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
MAOA P21397 1/20 0.36
DRD1 P21728 1/20 0.36
ACHE P22303 1/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7033840 0.83 MAPT (0.63) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL29847798 0.77 KDM4E (0.73) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL8806485 0.77 KDM4E (0.73) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL31289478 0.76 KDM4E (0.76) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL14447528 0.75 KDM4E (0.57) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL7033846 0.73 MAPT (0.82) KDM4EMAPTGFERRAB9AALDH1A1
Dimethylamine SCHEMBL16741824 0.72 KDM4E (0.68) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL22091286 0.68 MAPT (0.94) KDM4EMAPTGFERRAB9AALDH1A1
SCHEMBL22982922 0.67 PARP1 (0.56) KDM4EMAPTGFERSMN1; SMN2KMT2A
SCHEMBL31289521 0.67 MEN1 (0.56) KDM4EMAPTGFERRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3339305-B1 INDOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND USE THEREOF IN PHARMACEUTICAL DRUG ZHEJIANG HISUN PHARM CO LTD (CN) 2022-05-04 EP disclosed