SCHEMBL29501019

SCHEMBL29501019

COc1ccc([C@H]2C(CO)C(=O)N2c2cc(OC)c(OC)c(OC)c2)cc1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
HDAC1 Q13547 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
ESR1 P03372 3/20 0.45
ESR2 Q92731 2/20 0.45
SMPD1 P17405 1/20 0.44
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
APP P05067 2/20 0.43
ABCB1 P08183 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SOAT1 P35610 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30184680 1.00 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL29500979 1.00 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL28911331 0.90 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL20708020 0.90 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19423198 0.90 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19423057 0.90 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL20707978 0.88 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL19423000 0.88 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL30479081 0.86 TDP1 (0.44) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL24167129 0.86 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380728-A Novel diaryl-beta-lactam organic selenium compound, preparation method and application thereof in pharmacy 复旦大学 2022-04-22 CN disclosed