SCHEMBL29503147

SCHEMBL29503147

NC(=O)c1cccc(C(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.57
MAPT P10636 3/20 0.46
TSHR P16473 2/20 0.46
CYP3A4 P08684 2/20 0.46
RECQL P46063 2/20 0.46
PMP22 Q01453 2/20 0.46
HSD17B10 Q99714 2/20 0.46
POLB P06746 1/20 0.46
CYP2C19 P33261 1/20 0.46
BLM P54132 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PARP15 Q460N3 2/20 0.44
PARP10 Q53GL7 2/20 0.44
TNKS O95271 1/20 0.44
PARP14 Q460N5 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PTGS1 P23219 2/20 0.43
CXCR1 P25024 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13908477 1.00 PARP1 (0.57) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL28204633 0.85 PARP1 (0.53) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL84456 0.84 PARP1 (0.57) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL30154821 0.84 PARP1 (0.57) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL8249965 0.82 PARP1 (0.55) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL211856 0.82 PARP1 (0.55) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL8255364 0.82 PARP1 (0.55) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL12052133 0.82 PARP1 (0.55) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL1116685 0.82 PARP1 (0.50) PARP1MAPTTSHRCYP3A4RECQL
SCHEMBL315064 0.82 ANPEP (0.58) MAPTTSHRCYP3A4RECQLPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN claimed
CN-116715625-A Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-09-08 CN disclosed
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN disclosed