SCHEMBL29515487

SCHEMBL29515487

c1ccc2c(c1)ccn2CCCN1CCN(c2nsc3ccccc23)CC1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.60
HTR1A P08908 7/20 0.60
DRD2 P14416 7/20 0.60
ADRA1D P25100 2/20 0.60
ADRA1B P35368 2/20 0.60
HTR7 P34969 5/20 0.56
HTR6 P50406 5/20 0.56
SIGMAR1 Q99720 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8831833 0.82 HTR2A (0.67) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL8831311 0.80 HTR2A (0.70) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL8831370 0.80 HTR2A (0.66) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL25335774 0.80 HTR2A (0.67) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL30515499 0.80 HTR2A (0.67) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL8419556 0.79 HTR2A (0.67) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL8671981 0.78 HTR2A (0.65) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL6185115 0.78 HTR2A (0.65) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL792909 0.78 HTR2A (0.65) HTR2AHTR1ADRD2ADRA1DADRA1B
SCHEMBL7771353 0.78 HTR2A (0.65) HTR2AHTR1ADRD2ADRA1DADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109467554-B Indole-heteroaromatic piperazine (pyridine) derivative and application thereof in anti-depression 上海医药工业研究院 2022-05-10 CN claimed