SCHEMBL2953304

SCHEMBL2953304

CCC(C(=O)O)C1(O)CCN(Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.55
OPRL1 P41146 1/20 0.54
POLB P06746 1/20 0.52
ALDH1A1 P00352 3/20 0.52
CHRM2 P08172 3/20 0.50
CHRM3 P20309 2/20 0.50
CCR3 P51677 1/20 0.49
CYP3A4 P08684 4/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2C19 P33261 3/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
SIGMAR1 Q99720 1/20 0.47
USP2 O75604 1/20 0.47
MAPK1 P28482 1/20 0.47
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11374272 0.90 CYP2D6 (0.53) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL11370652 0.84 CYP2D6 (0.60) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL4485326 0.80 OPRL1 (0.61) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL18075917 0.80 CYP2D6 (0.55) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL11394628 0.79 CYP2D6 (0.56) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL23316097 0.78 CYP2D6 (0.53) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL29822404 0.78 CHRM2 (0.51) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL17101387 0.78 CHRM2 (0.51) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL1681535 0.78 CYP2D6 (0.56) CYP2D6OPRL1POLBALDH1A1CHRM2
SCHEMBL23744794 0.77 OPRL1 (0.61) CYP2D6OPRL1POLBALDH1A1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759340-B2 Antibacterial agents GLAXO GROUP LIMITED (GB) 2010-07-20 US disclosed
US-4255432-A ANTIHYPERTENSIVE AGENTS, ANTIHISTAMINES, BRONCHODILATOR AGENTS, ANTIVASOSPASTIC AGENTS SYNTEX (U.S.A.) INC. (US) 1981-03-10 US disclosed
US-4244961-A 1-Oxa-3,8-diazaspiro[4.5]decan-2-ones antihypertensive agents SYNTEX (U.S.A.) INC. (US) 1981-01-13 US disclosed