SCHEMBL29534445

SCHEMBL29534445

C=CC(=O)Nc1cccc(Oc2nc(Cl)ncc2Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.67
BTK Q06187 6/20 0.64
JAK2 O60674 2/20 0.61
BLK P51451 2/20 0.61
BMX P51813 2/20 0.61
JAK3 P52333 2/20 0.61
CTSC P53634 4/20 0.58
ITK Q08881 3/20 0.58
PLK4 O00444 1/20 0.55
GAK O14976 1/20 0.55
NUAK1 O60285 1/20 0.55
FLT3 P36888 1/20 0.55
PTK2 Q05397 1/20 0.55
ERBB4 Q15303 1/20 0.55
DCLK3 Q9C098 1/20 0.55
NUAK2 Q9H093 1/20 0.55
EML4 Q9HC35 1/20 0.55
EIF2AK4 Q9P2K8 1/20 0.55
ALK Q9UM73 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9945484 1.00 EGFR (0.67) EGFRBTKJAK2BLKBMX
SCHEMBL9945482 0.89 EGFR (0.57) EGFRBTKJAK2BLKBMX
SCHEMBL9946942 0.89 EGFR (0.67) EGFRBTKJAK2BLKBMX
SCHEMBL9945479 0.89 BTK (0.65) EGFRBTKJAK2BLKBMX
SCHEMBL16370708 0.89 EGFR (0.73) EGFRBTKCTSCITK
SCHEMBL16391074 0.87 EGFR (0.65) EGFRBTKJAK2BLKBMX
SCHEMBL9946937 0.86 EGFR (0.66) EGFRBTKITK
SCHEMBL21358332 0.83 EGFR (0.59) EGFRBTKJAK2BLKBMX
SCHEMBL23899138 0.81 MAP2K7 (0.59) EGFRBTKCTSCITK
SCHEMBL9924751 0.81 EGFR (0.72) EGFRBTKJAK2BLKBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111393377-B Deuterated pyrimidine derivative with anticancer effect 四川大学华西医院 2022-04-05 CN disclosed