Sulindac Sulfide

Sulindac Sulfide

SCHEMBL29536153

CSc1ccc(/C=C2/C(C)=C(CC(=O)O)c3cc(F)ccc32)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 14/20 1.00
CYP1A2 P05177 3/20 1.00
MAPT P10636 3/20 1.00
MAPK1 P28482 3/20 1.00
PTGS2 P35354 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
PTGS1 P23219 2/20 1.00
EGFR P00533 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
DRD1 P21728 1/20 1.00
OPRM1 P35372 1/20 1.00
PSEN1 P49768 1/20 1.00
PSEN2 P49810 1/20 1.00
APH1B Q8WW43 1/20 1.00
NCSTN Q92542 1/20 1.00
APH1A Q96BI3 1/20 1.00
PSENEN Q9NZ42 1/20 1.00
CYSLTR1 Q9Y271 1/20 1.00
PTGDR2 Q9Y5Y4 1/20 1.00
RXRA P19793 5/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulindac Sulfide SCHEMBL2221399 1.00 PPARG (1.00) PPARGCYP1A2MAPTMAPK1PTGS2
Sulindac Sulfide SCHEMBL4780668 1.00 PPARG (1.00) PPARGCYP1A2MAPTMAPK1PTGS2
Sulindac Sulfide SCHEMBL2586650 1.00 PPARG (1.00) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL15631472 0.91 PPARG (0.83) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL8149218 0.91 PPARG (0.83) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL24101275 0.91 PPARG (0.86) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL8149214 0.91 PPARG (0.83) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL8149223 0.91 PPARG (0.83) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL30486787 0.91 PPARG (0.86) PPARGCYP1A2MAPTMAPK1PTGS2
SCHEMBL22109319 0.90 PPARG (0.81) PPARGCYP1A2MAPTMAPK1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12419876-B2 Treatment of hearing loss by inhibition of casein kinase 1 MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2025-09-23 US disclosed
EP-3970725-B1 A GAMMA SECRETASE INHIBITOR FOR TREATING HEARING LOSS MASSACHUSETTS EYE & EAR INFIRMARY (US) 2025-08-20 EP disclosed
US-20250099539-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS MASSACHUSETTS EYE AND EAR INFIRMARY 2025-03-27 US disclosed
US-12239651-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2025-03-04 US disclosed
US-12161647-B2 Treating hearing loss MASSACHUSETTS EYE & EAR INFIRMARY (US) 2024-12-10 US disclosed
US-12156899-B2 Methods and compositions for regenerating hair cells and/or supporting cells MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-12-03 US disclosed
WO-2024218483-A1 SULINDAC AND/OR SULINDAC SULFIDE FOR THE TREATMENT OF ANGELMAN SYNDROME HEALX LTD (GB) 2024-10-24 WO disclosed
WO-2024218483-A1 SULINDAC AND/OR SULINDAC SULFIDE FOR THE TREATMENT OF ANGELMAN SYNDROME HEALX LTD (GB) 2024-10-24 WO disclosed
US-20240299432-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY 2024-09-12 US disclosed
US-12043653-B2 Efficient delivery of therapeutic molecules to cells of the inner ear MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-07-23 US disclosed
US-11963968-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2024-04-23 US disclosed
US-20230277574-A1 TREATMENT OF HEARING LOSS MASSACHUSETTS EYE AND EAR INFIRMARY 2023-09-07 US disclosed
CN-109689071-B Human airway stem cells in lung epithelial engineering 通用医疗公司 2023-05-30 CN disclosed
US-11590152-B2 Treatment of hearing loss MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2023-02-28 US disclosed
US-20220281941-A1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2022-09-08 US disclosed
US-11370823-B2 Efficient delivery of therapeutic molecules to cells of the inner ear MASSACHUSETTS EYE AND EAR INFIRMARY (US) 2022-06-28 US disclosed
EP-3970725-A1 A GAMMA SECRETASE INHIBITOR FOR TREATING HEARING LOSS Massachusetts Eye & Ear Infirmary (US) 2022-03-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11370823-B2 Efficient delivery of therapeutic molecules to cells of the inner ear HES1, NOTCH1, NOTCH2 PPARG 3372/4885CYP1A2 4807/4885MAPT 3320/4885
US-12419876-B2 Treatment of hearing loss by inhibition of casein kinase 1 GSK3B, GSKIP, BACE1 PPARG 4448/4885CYP1A2 4713/4885MAPT 1681/4885
US-20240299432-A1 TREATMENT OF HEARING LOSS HES1, NOTCH1, NOTCH4 PPARG 3326/4885CYP1A2 4835/4885MAPT 3170/4885
US-20220281941-A1 EFFICIENT DELIVERY OF THERAPEUTIC MOLECULES TO CELLS OF THE INNER EAR HES1, NOTCH1, NOTCH2 PPARG 3372/4885CYP1A2 4807/4885MAPT 3320/4885
US-11590152-B2 Treatment of hearing loss HES1, NOTCH1, NOTCH4 PPARG 3326/4885CYP1A2 4835/4885MAPT 3170/4885
US-12161647-B2 Treating hearing loss BACE1, BACE2, PSENEN PPARG 2526/4885CYP1A2 3678/4885MAPT 1900/4885
US-20230277574-A1 TREATMENT OF HEARING LOSS HES1, NOTCH1, NOTCH4 PPARG 3326/4885CYP1A2 4835/4885MAPT 3170/4885
US-12043653-B2 Efficient delivery of therapeutic molecules to cells of the inner ear HES1, NOTCH1, NOTCH2 PPARG 3372/4885CYP1A2 4807/4885MAPT 3320/4885
US-12156899-B2 Methods and compositions for regenerating hair cells and/or supporting cells HES1, NOTCH1, NOTCH4 PPARG 3963/4885CYP1A2 4810/4885MAPT 3747/4885
US-20250099539-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS AND/OR SUPPORTING CELLS HES1, NOTCH1, NOTCH4 PPARG 3963/4885CYP1A2 4810/4885MAPT 3747/4885
US-12239651-B2 Treatment of hearing loss HES1, NOTCH1, NOTCH4 PPARG 3326/4885CYP1A2 4835/4885MAPT 3170/4885
US-11963968-B2 Treatment of hearing loss HES1, NOTCH1, NOTCH4 PPARG 3326/4885CYP1A2 4835/4885MAPT 3170/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.