SCHEMBL2953709

SCHEMBL2953709

CC(CO[Si](C)(C)C(C)(C)C)Oc1cc(Oc2ccc(C(=O)N3CCC3)cc2F)cc(C(=O)Nc2nccs2)c1

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCK P35557 20/20 0.63
KCNH2 Q12809 5/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905733 1.00 GCK (0.63) GCKKCNH2
SCHEMBL2656429 0.90 GCK (0.78) GCKKCNH2
SCHEMBL2655069 0.89 GCK (0.80) GCKKCNH2
SCHEMBL3255054 0.88 GCK (0.65) GCKKCNH2
SCHEMBL1427050 0.88 GCK (0.65) GCKKCNH2
SCHEMBL2905305 0.87 GCK (0.63) GCKKCNH2
SCHEMBL4794169 0.87 GCK (0.63) GCKKCNH2
SCHEMBL2654209 0.85 GCK (0.65) GCKKCNH2
SCHEMBL1493733 0.85 GCK (0.65) GCKKCNH2
SCHEMBL1493734 0.85 GCK (0.65) GCKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756076-B1 HETROARYL BENZAMIDE DERIVATIVES FOR USE AS GLK ACTIVATORS IN THE TREATMENT OF DIABETES ASTRAZENECA AB (SE) 2010-08-11 EP disclosed