SCHEMBL29538495

SCHEMBL29538495

CN1CCN(c2ccc(-c3cc4c(Oc5cccc(CC#CCN)c5)ncnc4n3COCC[Si](C)(C)C)cc2)CC1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
USP2 O75604 2/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 2/20 0.31
CYP1A2 P05177 2/20 0.31
MAPK1 P28482 2/20 0.31
HIF1A Q16665 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
EGFR P00533 1/20 0.31
KIT P10721 1/20 0.31
FLT3 P36888 1/20 0.31
DGAT1 O75907 1/20 0.31
AOC3 Q16853 1/20 0.31
FYN P06241 1/20 0.30
PRMT5 O14744 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21484372 1.00 PIM1 (0.32) PIM1PIM3USP2ALDH1A1LMNA
SCHEMBL21484369 0.90 KIT (0.33) PIM1PIM3USP2MAPK1MAPKAPK2
SCHEMBL21484319 0.87 EGFR (0.39) PIM1PIM3USP2ALDH1A1LMNA
SCHEMBL21758097 0.80 EGFR (0.39) EGFR
SCHEMBL21484367 0.79 EGFR (0.51) EGFRFLT3
SCHEMBL29538509 0.78 JAK3 (0.46) EGFR
SCHEMBL21516142 0.78 EGFR (0.37) EGFR
SCHEMBL23035014 0.78 PRMT5 (0.51) KITPRMT5
SCHEMBL29538307 0.78 PRMT5 (0.51) KITPRMT5
SCHEMBL21484350 0.76 PIM1 (0.40) PIM1PIM3LMNAMAPKAPK2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110072865-B Pyrrolo-aromatic heterocyclic compounds, preparation method and medical application thereof 中国医药研究开发中心有限公司 2022-02-11 CN disclosed