SCHEMBL29544462

SCHEMBL29544462

COc1c(F)cccc1Nc1c(-c2ccncc2NC(=O)C2CCC2)nn2c1C(=O)NCC2

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 5/20 0.42
EGFR P00533 7/20 0.42
GSK3B P49841 3/20 0.38
GSK3A P49840 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29544947 0.97 TYK2 (0.45) TYK2EGFRGSK3BGSK3AADORA2A
SCHEMBL29545072 0.90 EGFR (0.42) TYK2EGFRGSK3BGSK3A
SCHEMBL29545071 0.90 EGFR (0.42) TYK2EGFRGSK3BGSK3A
SCHEMBL29545545 0.87 EGFR (0.45) TYK2EGFR
SCHEMBL29544404 0.87 EGFR (0.43) TYK2EGFR
SCHEMBL29544687 0.87 EGFR (0.43) TYK2EGFR
SCHEMBL29544823 0.87 EGFR (0.46) TYK2EGFR
SCHEMBL29545632 0.86 EGFR (0.46) TYK2EGFR
SCHEMBL29544852 0.85 EGFR (0.49) EGFR
SCHEMBL29544860 0.85 EGFR (0.49) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022072634-A1 BICYCLIC COMPOUNDS FOR USE IN THE TREATMENT CANCER SCORPION THERAPEUTICS, INC. (US) 2022-04-07 WO disclosed