SCHEMBL29555960

SCHEMBL29555960

CN(CCN1CCC(c2ccc3[nH]c(Br)c(CC4CC4)c3c2)CC1)C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 19/20 0.42
TLR9 Q9NR96 18/20 0.42
TLR8 Q9NR97 14/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19850077 1.00 TLR7 (0.42) TLR7TLR9TLR8HRH3
SCHEMBL19850120 0.92 TLR9 (0.46) TLR7TLR9TLR8
SCHEMBL29555861 0.92 TLR9 (0.46) TLR7TLR9TLR8
SCHEMBL19839197 0.88 TLR9 (0.44) TLR7TLR9TLR8HRH3
SCHEMBL19838429 0.82 TLR7 (0.47) TLR7TLR9TLR8
SCHEMBL19839243 0.79 TLR9 (0.50) TLR7TLR9TLR8
SCHEMBL19839198 0.78 TLR9 (0.49) TLR7TLR9TLR8
SCHEMBL4564154 0.78 HRH3 (0.43) TLR7TLR9HRH3
SCHEMBL5805849 0.77 HRH3 (0.45) HRH3
SCHEMBL19849996 0.76 TLR7 (0.69) TLR7TLR9TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715617-B Dimethoxyphenyl-substituted indole compounds as inhibitors of TLR7, TLR8 or TLR9 百时美施贵宝公司 2022-04-19 CN disclosed