SCHEMBL29563264

SCHEMBL29563264

O=C(O)CNC(=O)c1ncc(-c2ccc(F)c(Cl)c2)cc1O

nearest known ligand 0.76

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 19/20 0.76
EGLN3 Q9H6Z9 9/20 0.76
FLT1 P17948 7/20 0.71
VEGFA P15692 7/20 0.71
TET3 O43151 1/20 0.71
BBOX1 O75936 1/20 0.71
ASPH Q12797 1/20 0.71
TET2 Q6N021 1/20 0.71
KDM8 Q8N371 1/20 0.71
OGFOD1 Q8N543 1/20 0.71
TET1 Q8NFU7 1/20 0.71
HIF1AN Q9NWT6 1/20 0.71
FTO Q9C0B1 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920683 0.87 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL19933509 0.86 EGLN1 (0.72) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL1921949 0.84 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL19933464 0.84 EGLN1 (0.72) EGLN1EGLN3FLT1VEGFATET3
Vadadustat SCHEMBL29357486 0.83 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
Vadadustat SCHEMBL29405970 0.83 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
Vadadustat SCHEMBL1920738 0.83 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL29563907 0.83 EGLN1 (0.79) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL3484399 0.82 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3
SCHEMBL30145054 0.82 EGLN1 (1.00) EGLN1EGLN3FLT1VEGFATET3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022078428-A1 COMPOUND AS PROLYL HYDROXYLASE INHIBITOR AND PREPARATION METHOD THEREFOR 江苏苏中药业集团股份有限公司 2022-04-21 WO disclosed