SCHEMBL29564744

SCHEMBL29564744

CS(=O)(=O)NCCNC(=O)c1cccc(-n2ccc3cc(C(=O)N4CCC(F)(F)CC4)cnc32)c1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.49
IRAK4 Q9NWZ3 4/20 0.43
PTK2 Q05397 10/20 0.40
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23675326 1.00 HPGD (0.49) HPGDIRAK4PTK2MGLL
SCHEMBL23675155 0.91 HPGD (0.46) HPGDIRAK4MGLL
SCHEMBL29564963 0.89 HPGD (0.54) HPGDPTK2MGLL
SCHEMBL23675145 0.89 HPGD (0.54) HPGDPTK2MGLL
SCHEMBL23675235 0.88 HPGD (0.53) HPGDPTK2MGLL
SCHEMBL29673063 0.86 HPGD (0.48) HPGDPTK2MGLL
SCHEMBL28887253 0.86 HPGD (0.48) HPGDPTK2MGLL
SCHEMBL29565007 0.82 HPGD (0.57) HPGDPTK2MGLL
SCHEMBL23675325 0.82 HPGD (0.57) HPGDPTK2MGLL
SCHEMBL24942913 0.81 HPGD (0.61) HPGDMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115335043-B PGDH inhibitors and methods of making and using the same 迈欧伏特治疗公司 2025-03-28 CN disclosed
CN-117377668-A Inhalant formulations of PGDH inhibitors and methods of use thereof 迈欧伏特治疗公司 2024-01-09 CN disclosed
EP-4228650-A1 INHALED FORMULATIONS OF PGDH INHIBITORS AND METHODS OF USE THEREOF Epirium Bio Inc. (US) 2023-08-23 EP disclosed
EP-4093385-A1 PGDH INHIBITORS AND METHODS OF MAKING AND USING Myoforte Therapeutics Inc. (US) 2022-11-30 EP disclosed
CN-115335043-A PGDH inhibitors and methods of making and using 迈欧伏特治疗公司 2022-11-11 CN disclosed
WO-2022082009-A1 INHALED FORMULATIONS OF PGDH INHIBITORS AND METHODS OF USE THEREOF EPIRIUM BIO INC. (US) 2022-04-21 WO disclosed