SCHEMBL29565633

SCHEMBL29565633

CC1(N)C(=O)N(c2cc(Cc3n[nH]c(=O)c4ccccc34)ccn2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.51
AR P10275 1/20 0.45
TSHR P16473 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ENPP1 P22413 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24390020 1.00 PARP1 (0.51) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL25890809 0.90 PARP1 (0.50) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL29566305 0.90 PARP1 (0.49) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL25313203 0.89 PARP1 (0.49) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL25890293 0.89 PARP1 (0.49) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL29565612 0.85 PARP1 (0.62) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL24389992 0.85 PARP1 (0.62) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL29565753 0.84 PARP1 (0.45) PARP1ARTSHRCYP3A4CYP2C9
SCHEMBL24390012 0.83 PARP1 (0.70) PARP1TSHRCYP3A4CYP2C9CYP2C19
SCHEMBL29565339 0.83 PARP1 (0.70) PARP1TSHRCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022090938-A1 PHTHALAZINONE DERIVATIVES USEFUL AS PARP INHIBITORS RHIZEN PHARMACEUTICALS AG (CH) 2022-05-05 WO disclosed