SCHEMBL29592128

SCHEMBL29592128

O=C(Nc1cccc(F)c1)Nc1cc(F)c(F)c(C(=O)c2ccc3ncc(N4CCOCC4)nc3c2)c1F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.46
MTOR P42345 8/20 0.46
PIK3CD O00329 6/20 0.46
PIK3CG P48736 6/20 0.46
PIK3CB P42338 5/20 0.46
AKT1 P31749 1/20 0.44
HDAC3 O15379 2/20 0.41
HDAC2 Q92769 1/20 0.41
PRKDC P78527 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.41
DGAT1 O75907 1/20 0.41
EPHX2 P34913 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CDK6 Q00534 1/20 0.40
HPGD P15428 1/20 0.40
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14783938 1.00 PIK3CA (0.46) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL14783379 0.92 PIK3CA (0.46) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL29592442 0.92 PIK3CA (0.46) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL14783124 0.91 IDH2 (0.49) AKT1
SCHEMBL29590150 0.91 IDH2 (0.49) AKT1
SCHEMBL15619687 0.90 PIK3CA (0.44) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL14783129 0.90 PIK3CA (0.47) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL29590134 0.90 PIK3CA (0.47) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL15689190 0.90 PIK3CA (0.52) PIK3CAMTORPIK3CDPIK3CGPIK3CB
SCHEMBL14783980 0.89 PIK3CA (0.44) PIK3CAMTORPIK3CDPIK3CGPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403531-A Chemical entities, compositions, and methods as kinase inhibitors 润新生物公司 2022-11-29 CN disclosed
CN-108794411-B Certain chemical entities, compositions, and methods 润新生物公司 2022-06-07 CN disclosed