SCHEMBL29604199

SCHEMBL29604199

Fc1cccnc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
GABRG2 P18507 3/20 0.42
GABRB3 P28472 3/20 0.42
GABRA5 P31644 3/20 0.42
GABRA3 P34903 3/20 0.42
GABRA1 P14867 2/20 0.41
ALOX15 P16050 1/20 0.39
KDM4E B2RXH2 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAPK14 Q16539 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
DHODH Q02127 1/20 0.38
CYP2A6 P11509 1/20 0.38
TOP1 P11387 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2639667 1.00 FEN1 (0.43) FEN1TRPV1PTGS1PTGS2GABRG2
Pyridine SCHEMBL28163764 0.92 CYP2A6 (0.44) FEN1TRPV1PTGS1PTGS2GABRG2
SCHEMBL30211300 0.84 MAPK14 (0.53) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31517665 0.84 MAPK14 (0.53) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30007391 0.84 MAPK14 (0.53) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL15624391 0.83 TDP1 (0.44) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL4139478 0.81 SYK (0.47) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2843365 0.81 TRPV1 (0.43) FEN1TRPV1GABRG2GABRB3GABRA5
SCHEMBL28479998 0.81 TRPV1 (0.47) TRPV1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31306178 0.81 TRPV1 (0.43) FEN1TRPV1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3983074-A1 PYRIDINE CARBAMATES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS Janssen Pharmaceutica NV (BE) 2022-04-20 EP disclosed