SCHEMBL29614982

SCHEMBL29614982

Nc1ccc(-n2cccn2)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.52
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 1/20 0.47
TDO2 P48775 1/20 0.42
NLRP3 Q96P20 4/20 0.41
PCSK9 Q8NBP7 1/20 0.40
MPO P05164 1/20 0.39
TBK1 Q9UHD2 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
HDAC4 P56524 1/20 0.38
LMNA P02545 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA10 Q9GZZ6 1/20 0.38
CHRNA9 Q9UGM1 1/20 0.38
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17743393 1.00 NOTUM (0.52) NOTUMKDM4EALDH1A1MAPK1TDO2
SCHEMBL1953799 0.79 NOTUM (0.47) NOTUMKDM4EALDH1A1MAPK1TDO2
SCHEMBL18086479 0.78 NOTUM (0.52) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL30088437 0.78 NOTUM (0.52) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL27513112 0.78 NOTUM (0.61) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL23119642 0.78 NOTUM (0.52) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL23642208 0.78 NOTUM (0.52) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL31366246 0.78 NOTUM (0.61) NOTUMKDM4EALDH1A1MAPK1PCSK9
SCHEMBL23832369 0.77 PCSK9 (0.48) NOTUMKDM4EALDH1A1MAPK1NLRP3
SCHEMBL30088498 0.77 PCSK9 (0.48) NOTUMKDM4EALDH1A1MAPK1NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109803963-B Cyano-substituted heterocycles having USP30 inhibitor activity 特殊治疗有限公司 2022-04-26 CN disclosed