SCHEMBL29616628

SCHEMBL29616628

CC(C)(C)OC(=O)N1CC(C(=O)Nc2ccc(F)cc2Cl)C1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.55
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
USP30 Q70CQ3 2/20 0.47
POLB P06746 1/20 0.46
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN6 P29350 1/20 0.45
CHRM4 P08173 1/20 0.44
STS P08842 1/20 0.43
MAPT P10636 1/20 0.42
TP53 P04637 1/20 0.42
PARP1 P09874 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ABL1 P00519 1/20 0.42
RIN1 Q13671 1/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23149216 1.00 NTRK1 (0.55) NTRK1HDAC1HDAC2USP30POLB
SCHEMBL23648774 0.86 HDAC2 (0.50) NTRK1HDAC1HDAC2USP30POLB
SCHEMBL18138932 0.84 HDAC2 (0.50) NTRK1HDAC1HDAC2USP30POLB
SCHEMBL31158689 0.84 HDAC2 (0.50) NTRK1HDAC1HDAC2USP30POLB
SCHEMBL28778540 0.81 PTPN1 (0.63) HDAC1HDAC2PTPN2PTPN1PTPN6
SCHEMBL18208383 0.80 HPGD (0.48) NTRK1POLBCHRM4MAPTTP53
SCHEMBL18208382 0.80 HPGD (0.48) NTRK1POLBCHRM4MAPTTP53
SCHEMBL18138914 0.79 STS (0.49) NTRK1HDAC1HDAC2USP30PTPN2
SCHEMBL18464772 0.79 HSD17B10 (0.53) HDAC1HDAC2POLBPTPN2PTPN1
SCHEMBL22315433 0.78 NPSR1 (0.63) NTRK1USP30POLBNPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4034538-A1 NEW HETEROCYCLIC MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS F. Hoffmann-La Roche AG (CH) 2022-08-03 EP disclosed
CN-114401968-A Novel heterocyclic monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2022-04-26 CN disclosed