SCHEMBL29616982

SCHEMBL29616982

N#Cc1cncc(-c2nc(N)nc3c2cnn3Cc2ccc(N)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.45
ADORA1 P30542 14/20 0.45
HSP90AA1 P07900 1/20 0.41
TRAP1 Q12931 1/20 0.41
HDAC1 Q13547 4/20 0.41
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
ATM Q13315 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29616986 1.00 ADORA2A (0.45) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL23388283 1.00 ADORA2A (0.45) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL25549553 0.90 TLR7 (0.39) ADORA2AADORA1HDAC1KDM4EALDH1A1
SCHEMBL29944508 0.88 ADORA2A (0.60) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL29616988 0.88 ADORA2A (0.60) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL23388289 0.88 ADORA2A (0.60) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL23388364 0.88 ADORA2A (0.51) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL29616971 0.88 ADORA2A (0.51) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL23388284 0.87 ADORA2A (0.44) ADORA2AADORA1HSP90AA1TRAP1HDAC1
SCHEMBL29616994 0.87 ADORA2A (0.44) ADORA2AADORA1HSP90AA1TRAP1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425756-B Adenosine receptor antagonist compounds and uses thereof 日东制药株式会社 2025-05-13 CN disclosed
CN-114829363-B Adenosine receptor antagonist compounds 日东制药株式会社 2024-10-01 CN disclosed
EP-4061817-A1 ADENOSINE RECEPTOR ANTAGONIST COMPOUNDS Ildong Pharmaceutical Co., Ltd. (KR) 2022-09-28 EP disclosed
WO-2022107044-A1 PREVENTION AND/OR TREATMENT OF CNS DISORDERS ILDONG PHARMACEUTICAL CO., LTD. (KR) 2022-05-27 WO disclosed