SCHEMBL29617002

SCHEMBL29617002

Cc1cc(Cn2ncc3c(-c4cncc(C#N)c4)nc(N)nc32)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.44
ADORA1 P30542 13/20 0.44
ADORA3 P0DMS8 1/20 0.42
ADORA2B P29275 1/20 0.42
HDAC1 Q13547 4/20 0.40
HSP90AA1 P07900 1/20 0.39
TRAP1 Q12931 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29616994 1.00 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388284 1.00 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29617016 0.89 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29617022 0.89 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388312 0.89 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL29617020 0.89 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL23388313 0.88 ADORA2A (0.46) ADORA2AADORA1HDAC1HSP90AA1TRAP1
SCHEMBL29944186 0.88 ADORA2A (0.46) ADORA2AADORA1HDAC1HSP90AA1TRAP1
SCHEMBL29616983 0.88 ADORA2A (0.46) ADORA2AADORA1HDAC1HSP90AA1TRAP1
SCHEMBL23388283 0.87 ADORA2A (0.45) ADORA2AADORA1ADORA3ADORA2BHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116425756-B Adenosine receptor antagonist compounds and uses thereof 日东制药株式会社 2025-05-13 CN disclosed
CN-114829363-B Adenosine receptor antagonist compounds 日东制药株式会社 2024-10-01 CN disclosed
EP-4061817-A1 ADENOSINE RECEPTOR ANTAGONIST COMPOUNDS Ildong Pharmaceutical Co., Ltd. (KR) 2022-09-28 EP disclosed
WO-2022107044-A1 PREVENTION AND/OR TREATMENT OF CNS DISORDERS ILDONG PHARMACEUTICAL CO., LTD. (KR) 2022-05-27 WO disclosed