SCHEMBL29618073

SCHEMBL29618073

Clc1ncc(Br)c(-c2c[nH]c3ccccc23)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.52
CCNK O75909 1/20 0.52
CCNE1 P24864 1/20 0.52
CDK2 P24941 1/20 0.52
CDK9 P50750 1/20 0.52
CDK12 Q9NYV4 1/20 0.52
CLK1 P49759 2/20 0.49
CDK5 Q00535 2/20 0.49
CDK5R1 Q15078 2/20 0.49
RPS6KA5 O75582 1/20 0.49
PDGFRB P09619 2/20 0.46
TDO2 P48775 2/20 0.45
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
HTR5A P47898 1/20 0.45
PDGFRA P16234 1/20 0.45
HTT P42858 1/20 0.44
ALDH1A1 P00352 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517759 1.00 CCNT1 (0.52) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL29613520 0.85 RPS6KA5 (0.66) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL517461 0.85 RPS6KA5 (0.66) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL517438 0.83 JAK2 (0.55) CCNT1CCNKCDK9CDK12CLK1
SCHEMBL22510124 0.83 CDK5 (0.56) CLK1CDK5CDK5R1RPS6KA5PDGFRB
SCHEMBL23152046 0.83 CLK1 (0.71) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL518282 0.83 CDK5 (0.49) CLK1CDK5CDK5R1RPS6KA5PDGFRB
SCHEMBL24839575 0.83 CLK1 (0.71) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL30957423 0.83 CDK5 (0.49) CLK1CDK5CDK5R1RPS6KA5PDGFRB
SCHEMBL30687302 0.83 CLK1 (0.71) CCNT1CCNKCCNE1CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112292378-B Indole derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-06 CN disclosed
CN-116018141-A Salt and crystal form containing indole derivatives, and preparation method and application thereof 上海翰森生物医药科技有限公司 2023-04-25 CN disclosed
CN-114539226-A Crystal form containing indole derivative free base and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-05-27 CN disclosed