SCHEMBL29618370

SCHEMBL29618370

N#Cc1ccc2c(c1)C(F)(F)CC2

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.57
PNMT P11086 6/20 0.43
DRD2 P14416 4/20 0.43
DRD3 P35462 4/20 0.43
PDK2 Q15119 1/20 0.41
TRPA1 O75762 1/20 0.36
BACE1 P56817 3/20 0.36
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23782794 1.00 KDM1A (0.57) KDM1APNMTDRD2DRD3PDK2
SCHEMBL26892628 0.78 KDM1A (0.57) KDM1APNMTDRD2DRD3TRPA1
SCHEMBL23782971 0.77 KDM1A (0.53) KDM1APNMTDRD2DRD3PDK2
SCHEMBL29664282 0.74 KDM1A (0.53) KDM1APNMTDRD2DRD3PDK2
SCHEMBL26889683 0.74 KDM1A (0.53) KDM1APNMTDRD2DRD3TRPA1
SCHEMBL17987998 0.73 KDM1A (1.00) KDM1A
SCHEMBL19764445 0.73 KDM1A (0.72) KDM1APNMTDRD2DRD3BACE1
SCHEMBL23569863 0.71 KDM1A (0.40) KDM1ADRD2PDK2BACE1
SCHEMBL29741279 0.70 KDM1A (0.46) KDM1APNMTPDK2BACE1
SCHEMBL28942392 0.70 ESR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114591293-A Fused ring compound as Nav1.8 inhibitor and application thereof 成都康弘药业集团股份有限公司 2022-06-07 CN disclosed