SCHEMBL29620847

SCHEMBL29620847

CC(C)(C)c1ccc(-c2ccc(O)cc2NC(=O)c2c[nH]c3ccccc3c2=O)c(C(C)(C)C)c1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CFTR P13569 20/20 0.64
ADORA3 P0DMS8 1/20 0.64
ADRB3 P13945 1/20 0.64
TBXA2R P21731 1/20 0.64
SLC6A2 P23975 1/20 0.64
AGTR1 P30556 1/20 0.64
MC4R P32245 1/20 0.64
PTGS2 P35354 1/20 0.64
SLC6A3 Q01959 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11998126 0.87 CFTR (0.73) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL2035792 0.87 CFTR (0.77) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL398517 0.83 CFTR (0.70) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL18708392 0.81 CFTR (0.67) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL1732268 0.81 CFTR (0.70) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL397981 0.80 CFTR (0.69) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL29050127 0.79 CFTR (0.64) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL30492065 0.79 CFTR (0.64) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL397317 0.79 CFTR (0.73) CFTRADORA3ADRB3TBXA2RSLC6A2
Ivacaftor SCHEMBL351373 0.79 CFTR (1.00) CFTRADORA3ADRB3TBXA2RSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114380746-A Novel crystalline form of ivacaiton and preparation method thereof 台湾神隆股份有限公司 2022-04-22 CN disclosed