SCHEMBL29623554

SCHEMBL29623554

Oc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1O[C@H]1CCOC1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.70
ERBB2 P04626 2/20 0.65
EPHA2 P29317 1/20 0.64
KDR P35968 1/20 0.64
EPHB4 P54760 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL231729 1.00 EGFR (0.70) EGFRERBB2EPHA2KDREPHB4
SCHEMBL13606740 1.00 EGFR (0.70) EGFRERBB2EPHA2KDREPHB4
SCHEMBL185864 1.00 EGFR (0.70) EGFRERBB2EPHA2KDREPHB4
SCHEMBL5223991 0.96 EGFR (0.72) EGFRERBB2
SCHEMBL7219629 0.96 EGFR (0.72) EGFRERBB2
SCHEMBL1446628 0.95 EGFR (0.65) EGFRERBB2KDREPHB4
SCHEMBL4523013 0.93 EGFR (0.77) EGFRERBB2EPHA2KDREPHB4
SCHEMBL4523002 0.93 EGFR (0.77) EGFRERBB2EPHA2KDREPHB4
SCHEMBL13606791 0.93 EGFR (0.77) EGFRERBB2EPHA2KDREPHB4
SCHEMBL4524312 0.93 EGFR (0.77) EGFRERBB2EPHA2KDREPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110840847-B Pharmaceutical compositions for the treatment of cystic fibrosis transmembrane conductance regulator mediated diseases 沃泰克斯药物股份有限公司 2022-07-29 CN disclosed
CN-110713489-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-05-31 CN disclosed
CN-110183440-B Heteroaryl SYK inhibitors 勃林格殷格翰国际有限公司 2022-04-22 CN disclosed