SCHEMBL29624893

SCHEMBL29624893

COC(=O)c1nc2c(Br)c[nH]c2nc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.40
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 8/20 0.35
ALDH1A1 P00352 5/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
MAP2K1 Q02750 2/20 0.35
HPGD P15428 2/20 0.35
DAPK3 O43293 1/20 0.35
JAK2 O60674 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
ABL1 P00519 1/20 0.35
CSF1R P07333 1/20 0.35
RET P07949 1/20 0.35
MET P08581 1/20 0.35
PDGFRA P16234 1/20 0.35
PRKACA P17612 1/20 0.35
LTK P29376 1/20 0.35
GRK5 P34947 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20209204 1.00 NPSR1 (0.40) NPSR1MAPK1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20188999 0.83 NPSR1 (0.41) NPSR1MAPK1KDM4EALDH1A1SMN1; SMN2
SCHEMBL20189161 0.82 MAPK1 (0.41) NPSR1MAPK1KDM4EALDH1A1SMN1; SMN2
SCHEMBL29625123 0.82 NPSR1 (0.40) NPSR1KDM4EALDH1A1SMN1; SMN2MAP2K1
SCHEMBL20191162 0.82 NPSR1 (0.40) NPSR1KDM4EALDH1A1SMN1; SMN2MAP2K1
SCHEMBL30675211 0.74 NR4A2 (0.40) NPSR1MAPK1KDM4EL3MBTL1NR4A2
SCHEMBL21060003 0.74 NR4A2 (0.40) NPSR1MAPK1KDM4EL3MBTL1NR4A2
SCHEMBL20187674 0.73 MAPT (0.38) MAPK1
SCHEMBL28353230 0.71 NPSR1 (0.54) NPSR1KDM4EALDH1A1SMN1; SMN2MAP2K1
SCHEMBL14072998 0.70 NPSR1 (0.36) NPSR1MAPK1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110214141-B Benzodiazolium compounds as ENaC inhibitors 企业治疗学有限公司 2022-05-31 CN disclosed