SCHEMBL29628112

SCHEMBL29628112

CC#CC(=O)N1CC[C@@H](c2nc(-c3ccc(C(=O)Nc4ccccn4)cc3)n3c(N)nccc23)C1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.62
EGFR P00533 1/20 0.49
ERBB2 P04626 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
PTGS2 P35354 1/20 0.49
KDR P35968 1/20 0.49
TEC P42680 1/20 0.49
TXK P42681 1/20 0.49
BLK P51451 1/20 0.49
BMX P51813 1/20 0.49
JAK3 P52333 1/20 0.49
ITK Q08881 1/20 0.49
ERBB4 Q15303 1/20 0.49
GP6 Q9HCN6 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19877414 1.00 BTK (0.62) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877417 1.00 BTK (0.62) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877993 1.00 BTK (0.62) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877807 0.97 BTK (0.63) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877626 0.97 BTK (0.63) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877624 0.97 BTK (0.63) BTKEGFRERBB2ADORA3PTGS2
SCHEMBL19877777 0.91 BTK (0.55) BTK
SCHEMBL19877592 0.90 BTK (0.56) BTK
SCHEMBL19877763 0.90 BTK (0.50) BTK
SCHEMBL30167350 0.90 BTK (0.50) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4006035-A1 QUINAZOLINE DERIVATIVES AS TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF CANCER Neupharma, Inc. (US) 2022-06-01 EP disclosed