Gw305178X

Gw305178X

SCHEMBL29636843

NS(=O)(=O)c1ccc(N/N=C2\C(=O)Nc3ccc4ncccc4c32)cc1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.46
CA1 P00915 17/20 0.41
CA2 P00918 16/20 0.41
CA12 O43570 12/20 0.41
CA9 Q16790 12/20 0.41
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
KDR P35968 1/20 0.37
CA4 P22748 2/20 0.35
CA7 P43166 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gw305178X SCHEMBL5894133 1.00 EIF2AK2 (0.46) EIF2AK2CA1CA2CA12CA9
Gw305178X SCHEMBL5894138 1.00 EIF2AK2 (0.46) EIF2AK2CA1CA2CA12CA9
SCHEMBL12856312 0.83 EIF2AK2 (0.46) EIF2AK2CA1CA2CA12CA9
SCHEMBL5893985 0.81 CYP1A2 (0.35) CYP1A2
SCHEMBL5893988 0.81 CYP1A2 (0.35) CYP1A2
SCHEMBL5893496 0.79 EIF2AK2 (0.47) EIF2AK2CA1CA2CA12CA9
SCHEMBL5893487 0.79 EIF2AK2 (0.47) EIF2AK2CA1CA2CA12CA9
SCHEMBL6619758 0.79 EIF2AK2 (0.47) EIF2AK2CA1CA2CA12CA9
SCHEMBL12856344 0.79 EIF2AK2 (0.47) EIF2AK2CA1CA2CA12CA9
SCHEMBL5773570 0.78 CYP1A2 (0.48) MAPTALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220281930-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PATHOLOGICAL PAIN AND ITCH DUKE UNIVERSITY (US) 2022-09-08 US disclosed
EP-4017873-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PATHOLOGICAL PAIN AND ITCH Duke University (US) 2022-06-29 EP disclosed