SCHEMBL29639797

SCHEMBL29639797

CC#Cc1nnc(-c2cnc(OC)nc2OC)cc1[C@H]1C[C@@H]1C(C)C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.35
QPCT Q16769 1/20 0.31
QPCTL Q9NXS2 1/20 0.31
MDM2 Q00987 6/20 0.31
TP53 P04637 5/20 0.31
MTOR P42345 2/20 0.31
PIK3CD O00329 1/20 0.31
ABL1 P00519 1/20 0.31
EGFR P00533 1/20 0.31
HCK P08631 1/20 0.31
SRC P12931 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
EPHB4 P54760 1/20 0.31
PRKDC P78527 1/20 0.31
PI4KB Q9UBF8 1/20 0.31
ACP1 P24666 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24418244 1.00 NT5E (0.35) NT5EQPCTQPCTLMDM2TP53
SCHEMBL24418242 0.91 NT5E (0.36) NT5EQPCTQPCTL
SCHEMBL29639798 0.91 NT5E (0.36) NT5EQPCTQPCTL
SCHEMBL24418488 0.91 NT5E (0.36) NT5EQPCTQPCTL
SCHEMBL29467441 0.90 NT5E (0.36) NT5EQPCTQPCTLMDM2TP53
SCHEMBL28728598 0.90 NT5E (0.36) NT5EQPCTQPCTLMDM2TP53
SCHEMBL24514847 0.86 NT5E (0.39) NT5EQPCTQPCTLMDM2TP53
SCHEMBL29614342 0.86 NT5E (0.39) NT5EQPCTQPCTLMDM2TP53
SCHEMBL22869348 0.84 NT5E (0.49) NT5EQPCTQPCTLMDM2TP53
SCHEMBL22869335 0.84 NT5E (0.49) NT5EQPCTQPCTLMDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022095953-A1 PYRIDAZINE ALKYNE COMPOUNDS AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-12 WO disclosed
CN-114437038-A Pyridazine alkyne compound and application thereof 武汉人福创新药物研发中心有限公司 2022-05-06 CN disclosed