SCHEMBL29640940

SCHEMBL29640940

CS(=O)(=O)c1ncc2ccc(=O)n(C3CCCC3)c2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCND1 P24385 18/20 0.60
CDK2 P24941 18/20 0.60
CCNE1 P24864 16/20 0.60
CDK6 Q00534 12/20 0.60
CDK4 P11802 9/20 0.60
CCNT1 O60563 3/20 0.60
CDK9 P50750 3/20 0.60
CCND2 P30279 6/20 0.55
CCND3 P30281 6/20 0.55
CCNA2 P20248 4/20 0.55
FGFR1 P11362 1/20 0.55
FGFR2 P21802 1/20 0.55
FGFR4 P22455 1/20 0.55
FGFR3 P22607 1/20 0.55
CCNA1 P78396 3/20 0.52
CCNE2 O96020 2/20 0.49
PAK4 O96013 1/20 0.49
PAK1 Q13153 1/20 0.49
PKN1 Q16512 1/20 0.49
CCNB2 O95067 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19857389 1.00 CCND1 (0.60) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL29798894 0.87 CCNE1 (0.65) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL19863588 0.87 CCNE1 (0.65) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL29507679 0.86 CDK2 (0.48) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL22860376 0.84 CCNE1 (0.44) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL26758841 0.84 CCNE1 (0.61) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL26098023 0.81 CCNE1 (0.50) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL30312005 0.81 CCNE1 (0.50) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL24572618 0.80 CCNE1 (0.64) CCND1CDK2CCNE1CDK6CDK4
SCHEMBL29640946 0.80 CCNE1 (0.64) CCND1CDK2CCNE1CDK6CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4573094-A2 CDK2 INHIBITORS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2025-06-25 EP disclosed
CN-115702155-B Novel pyrido [2,3-d ] pyrimidin-7 (8H) -one derivatives 微境生物医药科技(上海)有限公司 2025-01-24 CN disclosed
US-20250018049-A1 COMPOUNDS FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEOSOME PATHWAY NIKANG THERAPEUTICS, INC. 2025-01-16 US disclosed
CN-114394966-B Pyridopyrimidinone CDK2/4/6 inhibitors 辉瑞公司 2024-10-11 CN disclosed
EP-4334307-A1 CDK2 DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2024-03-13 EP disclosed
WO-2024039903-A2 CDK2 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2024-02-22 WO disclosed
EP-4267575-A1 COMPOUNDS FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEOSOME PATHWAY Nikang Therapeutics, Inc. (US) 2023-11-01 EP disclosed
CN-116390921-A Heterocyclic compound with cyclin-dependent kinase inhibition activity, preparation method and medical application thereof 中国医药研究开发中心有限公司 2023-07-04 CN disclosed
CN-115702155-A Novel pyrido [2,3-d ] pyrimidin-7 (8H) -one derivatives 微境生物医药科技(上海)有限公司 2023-02-14 CN disclosed
WO-2022236058-A1 CDK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed
WO-2022140472-A1 COMPOUNDS FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEOSOME PATHWAY NIKANG THERAPEUTICS, INC. (US) 2022-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250018049-A1 COMPOUNDS FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PROTEOSOME PATHWAY CDK2, SKP2, CDK5 CCND1 125/4885CDK2 1/4885CCNE1 36/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.