SCHEMBL29642136

SCHEMBL29642136

N#Cc1cc(CO)ccc1Oc1cncc(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.52
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
SCN9A Q15858 1/20 0.42
VEGFA P15692 1/20 0.39
EPAS1 Q99814 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC22A12 Q96S37 2/20 0.39
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
CYP19A1 P11511 1/20 0.36
PLA2G7 Q13093 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875607 1.00 AR (0.52) ARCYP11B1CYP11B2SCN9AVEGFA
SCHEMBL875413 0.91 AR (0.43) ARCYP11B1CYP11B2SCN9AVEGFA
SCHEMBL24385793 0.85 CYP11B1 (0.41) ARCYP11B1CYP11B2SCN9AVEGFA
SCHEMBL14670094 0.84 AR (0.46) ARCYP11B1CYP11B2SCN9AVEGFA
SCHEMBL29918418 0.84 AR (0.60) ARSCN9A
SCHEMBL14656415 0.84 AR (0.60) ARSCN9A
SCHEMBL29769048 0.83 AR (0.57) ARSCN9AEPAS1SMN1; SMN2
SCHEMBL875321 0.83 AR (0.57) ARSCN9AEPAS1SMN1; SMN2
SCHEMBL875025 0.83 SLC22A12 (0.47) ARCYP11B1CYP11B2VEGFAEPAS1
SCHEMBL14661984 0.83 TLR8 (0.40) AREPAS1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3239135-B1 PYRIMIDONE COMPOUNDS USED AS LP-PLA2 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2022-05-04 EP disclosed