SCHEMBL29642969

SCHEMBL29642969

COC(=O)Nc1ccc2c(c1)CC(=O)N2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
TLK2 Q86UE8 1/20 0.53
CRBN Q96SW2 1/20 0.49
LRRK2 Q5S007 1/20 0.48
MAPKAPK2 P49137 1/20 0.48
AHR P35869 1/20 0.47
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2A Q12879 1/20 0.47
GRIN2B Q13224 1/20 0.47
GRIN2C Q14957 1/20 0.47
GRIN3A Q8TCU5 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10365651 0.87 CRBN (0.64) MEN1KMT2ACRBNHDAC3HDAC4
SCHEMBL2547584 0.86 SMYD3 (0.53) SMYD3TLK2CRBNLRRK2MAPKAPK2
SCHEMBL154971 0.85 SMYD3 (0.60) SMYD3TLK2CRBNLRRK2AHR
SCHEMBL155039 0.83 SMYD3 (0.53) SMYD3TLK2GRIN2DGRIN3BGRIN1
SCHEMBL29642948 0.83 SMYD3 (0.61) SMYD3TLK2CRBNLRRK2MAPKAPK2
SCHEMBL578342 0.83 SMYD3 (0.61) SMYD3TLK2CRBNLRRK2MAPKAPK2
SCHEMBL22425051 0.82 NPC1 (0.59) SMYD3MEN1KMT2ATLK2
SCHEMBL3171463 0.82 SMYD3 (0.60) SMYD3TLK2LRRK2AHRGRIN2D
SCHEMBL5728126 0.82 SMYD3 (0.64) SMYD3TLK2LRRK2MAPKAPK2AHR
SCHEMBL4405727 0.81 CRBN (0.65) SMYD3KMT2ATLK2CRBNLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed