SCHEMBL29645678

SCHEMBL29645678

CCn1cc(-c2nc3c4cccc(Cl)c4nc(N[C@@H]4CCCCNC4=O)n3n2)cn1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.35
ADORA2A P29274 6/20 0.34
ADORA1 P30542 6/20 0.34
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
TNF P01375 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
LITAF Q99732 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MKNK1 Q9BUB5 2/20 0.32
MKNK2 Q9HBH9 2/20 0.32
ADORA3 P0DMS8 5/20 0.32
ADORA2B P29275 4/20 0.32
MAPT P10636 2/20 0.32
THRB P10828 1/20 0.32
SCN9A Q15858 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979137 1.00 PIM1 (0.35) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL29648877 0.91 PIM1 (0.35) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL22978999 0.91 PIM1 (0.35) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL22988433 0.91 PIM1 (0.35) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL31149998 0.91 PIM1 (0.35) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL29645871 0.91 ADORA2A (0.37) ADORA2AADORA1MKNK1MKNK2ADORA3
SCHEMBL22980138 0.91 ADORA2A (0.37) ADORA2AADORA1MKNK1MKNK2ADORA3
SCHEMBL22980792 0.90 ADORA2A (0.39) ADORA2AADORA1TNFLITAFHSP90AB1
SCHEMBL22979685 0.90 PIM1 (0.34) PIM1ADORA2AADORA1PIM3PIM2
SCHEMBL22979003 0.89 PIM1 (0.34) PIM1ADORA2AADORA1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN claimed
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP claimed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed