SCHEMBL29646142

SCHEMBL29646142

O=C1NCCCC[C@H]1Nc1nc2c(Cl)cccc2c2nc(-c3cnn(C4CC4)c3)nn12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 6/20 0.33
ADORA2A P29274 4/20 0.33
ADORA1 P30542 4/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP3A5 P20815 2/20 0.33
CYP3A7 P24462 2/20 0.33
CYP2C19 P33261 2/20 0.33
PDK4 Q16654 2/20 0.33
CYP3A43 Q9HB55 2/20 0.33
MKNK1 Q9BUB5 2/20 0.33
MKNK2 Q9HBH9 2/20 0.33
PAK4 O96013 3/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
IRAK1 P51617 2/20 0.32
ADORA3 P0DMS8 3/20 0.31
ADORA2B P29275 3/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979183 1.00 PAK1 (0.33) PAK1ADORA2AADORA1CYP1A2CYP3A4
SCHEMBL22980138 0.91 ADORA2A (0.37) ADORA2AADORA1MKNK1MKNK2ADORA3
SCHEMBL29645871 0.91 ADORA2A (0.37) ADORA2AADORA1MKNK1MKNK2ADORA3
SCHEMBL29646077 0.90 PAK1 (0.34) PAK1CYP1A2CYP3A4CYP3A5CYP3A7
SCHEMBL22979075 0.90 PAK1 (0.34) PAK1CYP1A2CYP3A4CYP3A5CYP3A7
SCHEMBL22979395 0.89 HDAC1 (0.35) ADORA2AADORA1CYP1A2CYP3A4CYP3A5
SCHEMBL22979232 0.89 KDM5A (0.36) PAK1ADORA2AADORA1CYP1A2CYP3A4
SCHEMBL22980020 0.89 ADORA2A (0.38) PAK1ADORA2AADORA1
SCHEMBL22979892 0.88 ADORA2A (0.33) ADORA2AADORA1CYP1A2CYP3A4CYP3A5
SCHEMBL22979811 0.88 ADORA2A (0.34) ADORA2AADORA1MKNK1MKNK2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN claimed
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP claimed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed