SCHEMBL29654232

SCHEMBL29654232

Fc1cccc(Nc2nc(-c3nc(-c4cccnc4)cs3)cs2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 11/20 1.00
CYP1A2 P05177 11/20 1.00
CYP1B1 Q16678 11/20 1.00
MEN1 O00255 8/20 0.67
KMT2A Q03164 8/20 0.67
RAB9A P51151 5/20 0.67
MAPT P10636 3/20 0.67
SMN1; SMN2 Q16637 2/20 0.67
NPC1 O15118 5/20 0.67
PKM P14618 1/20 0.67
ALDH1A1 P00352 1/20 0.67
MAPK1 P28482 1/20 0.66
CASP3 P42574 1/20 0.60
SENP8 Q96LD8 1/20 0.60
SENP7 Q9BQF6 1/20 0.60
SENP6 Q9GZR1 1/20 0.60
LMNA P02545 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28936800 1.00 CYP1A1 (1.00) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL29654026 0.89 CYP1B1 (1.00) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL28716326 0.89 CYP1B1 (1.00) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL29654126 0.87 CYP1B1 (1.00) CYP1A1CYP1A2CYP1B1
SCHEMBL28707148 0.87 CYP1B1 (1.00) CYP1A1CYP1A2CYP1B1
SCHEMBL29654082 0.87 MEN1 (0.89) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL28712438 0.87 MEN1 (0.89) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL7540052 0.86 MAPK1 (0.84) CYP1A1CYP1A2CYP1B1MEN1KMT2A
SCHEMBL5025363 0.85 MAPT (0.74) CYP1A1CYP1A2CYP1B1MEN1KMT2A
Bromide SCHEMBL7691671 0.84 MAPK1 (0.82) CYP1A1CYP1A2CYP1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed