SCHEMBL29655149

SCHEMBL29655149

O=c1[nH]nc(Cc2ccc(F)c(Br)c2)c2cc(C(F)(F)F)ccc12

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.59
TNKS O95271 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
MAPT P10636 1/20 0.45
ENPP1 P22413 2/20 0.44
LMNA P02545 1/20 0.44
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19748946 1.00 PARP1 (0.59) PARP1TNKSTNKS2MAPTENPP1
SCHEMBL29655259 0.85 PARP1 (0.64) PARP1ENPP1LMNA
SCHEMBL19748474 0.85 PARP1 (0.64) PARP1ENPP1LMNA
SCHEMBL19747669 0.84 PARP1 (0.63) PARP1ENPP1LMNA
SCHEMBL29655088 0.84 PARP1 (0.63) PARP1ENPP1LMNA
SCHEMBL29483966 0.84 PARP1 (0.72) PARP1ENPP1LMNA
SCHEMBL4572876 0.84 PARP1 (0.72) PARP1ENPP1LMNA
SCHEMBL19748607 0.84 PARP1 (0.68) PARP1ENPP1LMNA
SCHEMBL29655224 0.84 PARP1 (0.68) PARP1ENPP1LMNA
SCHEMBL29654940 0.83 PARP1 (0.61) PARP1ENPP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843874-B Phthalazine derivatives useful as inhibitors of PARP1, PARP2 and/or tubulin for the treatment of cancer 加利福尼亚大学董事会 2022-05-27 CN disclosed