SCHEMBL29664306

SCHEMBL29664306

Cc1nc(Cl)c2cc3c(cnn3CCOCc3ccccc3)cc2n1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
BRD4 O60885 1/20 0.35
RECQL P46063 1/20 0.35
KCNH2 Q12809 3/20 0.35
MCHR1 Q99705 3/20 0.35
GPR39 O43194 1/20 0.34
MAPK1 P28482 1/20 0.34
NR3C1 P04150 1/20 0.34
DHODH Q02127 2/20 0.33
ERBB2 P04626 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
CYP3A4 P08684 1/20 0.33
PDE1C Q14123 1/20 0.33
USP2 O75604 1/20 0.33
RAB9A P51151 1/20 0.33
RHEB Q15382 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29047123 1.00 CYP1A2 (0.36) CYP1A2CYP2D6CYP2C19BRD4RECQL
SCHEMBL29664247 0.81 KDM4E (0.47) BRD4KCNH2MCHR1GPR39USP2
SCHEMBL29047115 0.81 KDM4E (0.47) BRD4KCNH2MCHR1GPR39USP2
SCHEMBL29047116 0.69 TLR8 (0.41) CYP1A2MCHR1MAPK1NR3C1TLR8
SCHEMBL29047119 0.66 GAA (0.39) MCHR1MAPK1PDE1C
SCHEMBL856542 0.66 CYP3A4 (0.52) CYP3A4RAB9A
SCHEMBL20509231 0.65 ELANE (0.55) TLR7
SCHEMBL21248471 0.65 TSHR (0.42) CYP1A2CYP2D6CYP2C19NR3C1
SCHEMBL21265213 0.65 TSHR (0.42) CYP1A2CYP2D6CYP2C19NR3C1RAB9A
SCHEMBL21248131 0.64 CYP1A2 (0.42) CYP1A2CYP2D6CYP2C19NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022121813-A1 SOS1 INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF 北京泰德制药股份有限公司 2022-06-16 WO disclosed