SCHEMBL29675894

SCHEMBL29675894

CC(=O)NC(C)(C)c1ccc2c(c1)OCCO2

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2C19 P33261 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
MAPT P10636 2/20 0.51
TRPV1 Q8NER1 7/20 0.48
KDM4E B2RXH2 2/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
MTOR P42345 1/20 0.46
KMT2A Q03164 1/20 0.46
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
ATM Q13315 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19469482 0.77 PTGS1 (0.49) CYP1A2CYP2C19NPSR1MAPTTRPV1
SCHEMBL27254652 0.76 ACACB (0.54) CYP1A2CYP2C19MAPTRAB9ANPC1
SCHEMBL22839330 0.75 POLB (0.44) CYP1A2CYP2C19NPSR1MAPTTRPV1
SCHEMBL84835 0.75 TRPV1 (0.49) MAPTTRPV1RAB9ASMN1; SMN2MEN1
SCHEMBL1900108 0.73 GAA (0.57) MAPTKDM4ETSHRGAALMNA
SCHEMBL23052641 0.72 MAPT (0.41) CYP1A2CYP2C19NPSR1MAPTTRPV1
SCHEMBL14349287 0.72 MAPT (0.41) CYP1A2CYP2C19NPSR1MAPTTRPV1
SCHEMBL29337534 0.72 MAPT (0.44) CYP1A2CYP2C19NPSR1MAPTTRPV1
SCHEMBL5861384 0.71 CYP1A2 (1.00) CYP1A2CYP2C19NPSR1MAPTKDM4E
SCHEMBL2607670 0.71 MAPT (0.63) CYP1A2CYP2C19NPSR1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108617166-B Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-05-17 CN claimed