SCHEMBL29699198

SCHEMBL29699198

CCCCc1cccc2c1C(=O)NC2=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 6/20 0.43
CTSG P08311 4/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
GSK3B P49841 1/20 0.41
PTPRB P23467 1/20 0.39
PARP1 P09874 1/20 0.39
CASP3 P42574 2/20 0.38
CASP2 P42575 1/20 0.36
CASP7 P55210 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
CTRC Q99895 1/20 0.36
BID P55957 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166776 1.00 ELANE (0.43) ELANECTSGKDM4EALDH1A1GAA
Hydrochloric Acid SCHEMBL27668518 0.98 ELANE (0.43) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL2508510 0.95 NR1H2 (0.47) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL29699286 0.95 NR1H2 (0.47) ELANECTSGKDM4EALDH1A1GAA
Bicarbonate SCHEMBL29212760 0.94 KDM4E (0.46) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL10725524 0.94 NR1H2 (0.49) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL8684492 0.94 NR1H2 (0.49) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL10730459 0.94 NR1H2 (0.49) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL10725242 0.94 NR1H2 (0.49) ELANECTSGKDM4EALDH1A1GAA
SCHEMBL9402093 0.94 NR1H2 (0.49) ELANECTSGKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527179-B Chain hydrocarbon substituted isoindoline-1, 3-diketone PDE4 inhibitor and pharmaceutical application thereof 苏州璞正医药有限公司 2023-07-07 CN disclosed
WO-2023015944-A1 SUBSTITUTED ISOINDOLIN-1,3-DIONE PDE4 INHIBITOR AND PHARMACEUTICAL USE THEREOF 苏州璞正医药有限公司 2023-02-16 WO disclosed
CN-114790164-B Substituted isoindoline-1,3-diketone PDE4 inhibitor and pharmaceutical application thereof 苏州璞正医药有限公司 2022-12-27 CN disclosed
CN-114790164-A Substituted isoindoline-1, 3-diketone PDE4 inhibitor and pharmaceutical application thereof 苏州璞正医药有限公司 2022-07-26 CN disclosed