SCHEMBL29699807

SCHEMBL29699807

O=c1oc(-c2ccccc2F)nc2sc3c(c12)CCCC3

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.73
ALDH1A1 P00352 7/20 0.73
HPGD P15428 6/20 0.73
KDM4E B2RXH2 5/20 0.73
CASP3 P42574 3/20 0.73
SENP7 Q9BQF6 2/20 0.73
SENP6 Q9GZR1 2/20 0.73
SMN1; SMN2 Q16637 9/20 0.70
RAB9A P51151 6/20 0.70
NFKB1 P19838 1/20 0.70
NFKB2 Q00653 1/20 0.70
RELA Q04206 1/20 0.70
KMT2A Q03164 6/20 0.67
MEN1 O00255 3/20 0.67
L3MBTL1 Q9Y468 2/20 0.67
POLB P06746 2/20 0.67
PLA2G1B P04054 1/20 0.67
BLM P54132 1/20 0.67
CASP6 P55212 1/20 0.67
CASP8 Q14790 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL914044 1.00 MAPT (0.73) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL914357 0.87 MAPT (0.74) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL913664 0.85 MAPT (0.71) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL914596 0.83 MAPT (0.77) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL913332 0.83 MAPT (0.72) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL912737 0.83 SMN1; SMN2 (1.00) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL913600 0.80 SMN1; SMN2 (1.00) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL914037 0.78 SMN1; SMN2 (0.77) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL20545354 0.77 SMN1; SMN2 (1.00) MAPTALDH1A1HPGDKDM4ECASP3
SCHEMBL912689 0.77 SMN1; SMN2 (1.00) MAPTALDH1A1HPGDKDM4ECASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114615984-B Benzoxazinone compounds as dual KLK5/7 inhibitors 分子皮肤治疗公司 2025-02-07 CN disclosed
EP-4037687-A1 BENZOXAZINONE COMPOUNDS AS KLK5/7 DUAL INHIBITORS Molecular Skin Therapeutics, Inc. (US) 2022-08-10 EP disclosed
CN-114615984-A Benzoxazinone compounds as KLK5/7 dual inhibitors 分子皮肤治疗公司 2022-06-10 CN disclosed