SCHEMBL29756286

SCHEMBL29756286

O=C(c1ccc(-c2ccc3ncc(C#Cc4ccc(O)nc4)n3n2)cc1)N1CCOCC1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 16/20 0.64
MKNK2 Q9HBH9 16/20 0.64
EIF4E P06730 8/20 0.55
CYP3A4 P08684 1/20 0.51
MTOR P42345 1/20 0.45
KCNH2 Q12809 2/20 0.43
HPGD P15428 1/20 0.42
GRM5 P41594 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16621118 1.00 MKNK1 (0.64) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL16620305 0.90 MKNK1 (0.63) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL29756278 0.90 MKNK1 (0.63) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL16626002 0.88 MKNK1 (0.61) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL16620849 0.88 MKNK1 (0.79) MKNK1MKNK2EIF4ECYP3A4KCNH2
SCHEMBL16620738 0.88 MKNK1 (0.60) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL29756323 0.88 MKNK1 (0.60) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL16621478 0.87 MKNK1 (0.64) MKNK1MKNK2EIF4ECYP3A4KCNH2
SCHEMBL16621031 0.87 MKNK1 (0.59) MKNK1MKNK2EIF4ECYP3A4MTOR
SCHEMBL16621224 0.85 MKNK1 (0.61) MKNK1MKNK2EIF4ECYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052501-B1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY SCIENCE TECH & RES (SG) 2022-06-22 EP disclosed