SCHEMBL29763550

SCHEMBL29763550

Cn1ccnc1C(=O)Nc1ccc(C(=O)N2CCNCC2)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 4/20 0.52
GRM4 Q14833 5/20 0.51
PTK6 Q13882 8/20 0.49
LCK P06239 2/20 0.46
AURKB Q96GD4 2/20 0.46
CDK8 P49336 2/20 0.46
ROCK1 Q13464 2/20 0.46
CHEK1 O14757 1/20 0.46
AURKA O14965 1/20 0.46
DAPK3 O43293 1/20 0.46
JAK2 O60674 1/20 0.46
PRKD3 O94806 1/20 0.46
PAK4 O96013 1/20 0.46
ABL1 P00519 1/20 0.46
NTRK1 P04629 1/20 0.46
FYN P06241 1/20 0.46
CSF1R P07333 1/20 0.46
RET P07949 1/20 0.46
IGF1R P08069 1/20 0.46
MET P08581 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30581371 0.92 GRM1 (0.46) GRM1GRM4PTK6LCKAURKB
SCHEMBL30098796 0.90 GRM1 (0.47) GRM1GRM4PTK6LCKAURKB
SCHEMBL30581385 0.88 GRM1 (0.46) GRM1GRM4PTK6LCKAURKB
SCHEMBL30581370 0.83 GRM1 (0.44) GRM1GRM4PTK6LCKAURKB
SCHEMBL29437653 0.83 GRM1 (0.42) GRM1GRM4PTK6NAMPTCBLB
SCHEMBL30581367 0.83 GRM1 (0.48) GRM1GRM4PTK6NAMPT
SCHEMBL30581373 0.82 GRM4 (0.46) GRM1GRM4PTK6ROCK1JAK3
SCHEMBL22405623 0.82 LCK (0.47) PTK6LCKAURKBCDK8ROCK1
SCHEMBL29402806 0.82 LCK (0.47) PTK6LCKAURKBCDK8ROCK1
Hydrochloric Acid SCHEMBL22405648 0.81 LCK (0.46) PTK6LCKAURKBCDK8ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4288424-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-12-13 EP disclosed
WO-2022167631-A1 NOVEL HETEROARYL-SUBSTITUTED IMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2022-08-11 WO disclosed