Olsalazine

Olsalazine

SCHEMBL29769

O=C(O)c1cc(N=Nc2ccc(O)c(C(=O)O)c2)ccc1O.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ALOX5PPARGPTGS1PTGS2

The experimentally established mechanism targets of Olsalazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 3/20 0.70
PTGS1 known ✓ P23219 1/20 0.70
ALOX5 known ✓ P09917 1/20 0.57
MEN1 O00255 3/20 0.96
KMT2A Q03164 3/20 0.96
KDR P35968 2/20 0.96
PDE4A P27815 1/20 0.96
BLVRB P30043 1/20 0.96
HTT P42858 1/20 0.96
TDP1 Q9NUW8 4/20 0.82
THRB P10828 2/20 0.82
RECQL P46063 2/20 0.82
APP P05067 1/20 0.82
BLM P54132 1/20 0.82
PHLPP2 Q6ZVD8 4/20 0.70
ALDH1A1 P00352 3/20 0.70
CYP2C9 P11712 2/20 0.70
HSD17B10 Q99714 2/20 0.70
CYP2C19 P33261 2/20 0.70
CYP2D6 P10635 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Olsalazine SCHEMBL19693100 1.00 MEN1 (0.96) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL2228872 1.00 MEN1 (0.96) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL2628413 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL29861404 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL25118 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL25119 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL29385751 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL29378994 0.98 MEN1 (1.00) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL5922630 0.96 MEN1 (0.96) MEN1KMT2AKDRPDE4ABLVRB
Olsalazine SCHEMBL28138401 0.96 MEN1 (0.96) MEN1KMT2AKDRPDE4ABLVRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3953 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567554-B Gel factor and hydrogel loaded with anti-inflammatory agent as well as preparation methods and application thereof 中国科学技术大学 2025-03-07 CN claimed
CN-118286469-B Preparation method for nonmetallic organic magnetic resonance nano diagnosis and treatment agent 中山大学·深圳 2024-12-20 CN claimed
WO-2024234393-A1 FLEXIBLE INTELLIGENT WOOD HAVING RESPONSE FUNCTION, ACTUATOR, AND MANUFACTURING METHOD 南京林业大学 2024-11-21 WO claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-118286469-A Preparation method for nonmetallic organic magnetic resonance nano diagnosis and treatment agent 中山大学·深圳 2024-07-05 CN claimed
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
CN-117567554-A Gel factor and hydrogel loaded with anti-inflammatory agent as well as preparation methods and application thereof 中国科学技术大学 2024-02-20 CN claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
CN-217865037-U Encapsulation equipment is used in production of olsalazine sodium capsule 南京爱文医药研发有限公司 2022-11-22 CN claimed
CN-217864869-U Powder metering device is used in production of olsalazine sodium capsule 南京爱文医药研发有限公司 2022-11-22 CN claimed
EP-1384479-A1 Preventing or reducing photosensitivity and/or phototoxicity reactions to antiinfective medications G.D. SEARLE & CO. (US) 2004-01-28 EP claimed
WO-2003088811-A2 GELSOLIN AS A PROGNOSTIC MARKER OF ARTHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-10-30 WO claimed
US-20030152566-A1 Soluble CD40L (CD154) as a prognostic marker of atherosclerotic diseases THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-08-14 US claimed
WO-2003040691-A2 SOLUBLE CD40L(CD154) AS A PROGNOSTIC MARKER OF ATHEROSCLEROTIC DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2003-05-15 WO claimed
JP-2001525058-A 2001-12-04 JP claimed
EP-1003501-A4 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM & WOMENS HOSPITAL (US) 2001-01-17 EP claimed
EP-1003501-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2000-05-31 EP claimed
WO-1998043630-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 1998-10-08 WO claimed
EP-0741570-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1996-11-13 EP claimed
WO-1995020387-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1995-08-03 WO claimed