SCHEMBL29786707

SCHEMBL29786707

O=C1C(=Cc2ccccc2F)CNCC1=Cc1ccccc1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 1.00
DYRK2 Q92630 3/20 1.00
RAF1 P04049 2/20 1.00
RPS6KB1 P23443 2/20 1.00
MAPK1 P28482 2/20 1.00
AKT1 P31749 2/20 1.00
AKT2 P31751 2/20 1.00
KDR P35968 2/20 1.00
PRKAG1 P54619 2/20 1.00
MAP2K1 Q02750 2/20 1.00
PRKAA1 Q13131 2/20 1.00
MAPK14 Q16539 2/20 1.00
NEK1 Q96PY6 2/20 1.00
PRKAB1 Q9Y478 2/20 1.00
ACHE P22303 1/20 0.54
FGFR1 P11362 1/20 0.51
IGF1R P08069 1/20 0.50
EGFR P00533 1/20 0.49
MAPKAPK2 P49137 1/20 0.49
PRDX1 Q06830 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1325644 1.00 IKBKB (1.00) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL30593591 1.00 IKBKB (1.00) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL1325643 1.00 IKBKB (1.00) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL29363457 1.00 IKBKB (1.00) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL8119310 1.00 IKBKB (1.00) IKBKBDYRK2RAF1RPS6KB1MAPK1
Hydrochloric Acid SCHEMBL29359400 0.98 IKBKB (0.96) IKBKBDYRK2RAF1RPS6KB1MAPK1
Acetic Acid SCHEMBL3187366 0.91 IKBKB (0.82) IKBKBDYRK2RAF1RPS6KB1MAPK1
Acetic Acid SCHEMBL3187370 0.91 IKBKB (0.82) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL17300373 0.81 IKBKB (0.67) IKBKBDYRK2RAF1RPS6KB1MAPK1
SCHEMBL8128818 0.80 IKBKB (0.67) IKBKBDYRK2RAF1RPS6KB1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117503764-A Application of curcumin analogue EF24 in preparation of medicines for treating idiopathic pulmonary fibrosis 中国科学院昆明动物研究所 2024-02-06 CN disclosed
CN-115232068-B Compound and preparation method and application thereof 北京中医药大学 2023-09-08 CN disclosed
CN-108191751-B 4-fluorobenzenesulfonyl substituted 3, 5-diarylmethylene-4-piperidone compound and preparation method thereof 滨州医学院 2023-06-27 CN disclosed
CN-108997310-B Asymmetric 3-pyridine substituted 3, 5-diarylmethylene-4-piperidone and preparation method thereof 滨州医学院 2023-06-27 CN disclosed
CN-108191750-B 3, 5-diarylmethylene-N-benzenesulfonyl-4-piperidone compound and preparation method thereof 滨州医学院 2023-06-27 CN disclosed
CN-108191742-B 4-acetamidobenzenesulfonyl-substituted 3, 5-diarylmethylene-4-piperidone compound and preparation method thereof 滨州医学院 2023-06-27 CN disclosed
CN-108997311-B Asymmetric 4-pyridine substituted 3, 5-diarylmethylene-4-piperidone and preparation method thereof 滨州医学院 2023-06-23 CN disclosed
CN-115232068-A Compound and preparation method and application thereof 北京中医药大学 2022-10-25 CN disclosed
CN-109053565-B N-benzenesulfonyl substituted asymmetric pyridine-piperidone compounds and preparation method thereof 滨州医学院 2022-08-12 CN disclosed
CN-109053564-B N-benzenesulfonyl substituted asymmetric piperidone compounds and preparation method thereof 滨州医学院 2022-05-24 CN disclosed