SCHEMBL29790963

SCHEMBL29790963

Cc1cc(=O)oc2cc(NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CCCNC(=N)N)ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA9 Q16790 2/20 0.44
KDM4E B2RXH2 6/20 0.43
ALDH1A1 P00352 6/20 0.43
HPGD P15428 5/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPY4R P50391 6/20 0.43
NPY1R P25929 5/20 0.43
NPY2R P49146 4/20 0.43
NPY5R Q15761 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
GAA P10253 2/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31045724 1.00 CA12 (0.44) CA12CA1CA9KDM4EALDH1A1
SCHEMBL31045822 0.96 KDM4E (0.45) CA12CA1CA9KDM4EALDH1A1
SCHEMBL30619377 0.96 KDM4E (0.45) CA12CA1CA9KDM4EALDH1A1
SCHEMBL29543910 0.96 CA12 (0.47) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7208685 0.96 CA12 (0.47) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7208677 0.96 CA12 (0.47) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7204719 0.95 KDM4E (0.48) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7204729 0.95 KDM4E (0.48) CA12CA1CA9KDM4EALDH1A1
SCHEMBL8499114 0.95 KDM4E (0.48) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7205674 0.92 CA12 (0.52) CA12CA1CA9KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022178128-A1 SELECTIVE NEUTRAL PH INHIBITOR OF CATHEPSIN B THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-25 WO disclosed