SCHEMBL29794866

SCHEMBL29794866

OC1CCN(c2ncc(-c3ccc4nc5n(c4n3)C(c3ccccc3)COC5)cn2)CC1(F)F

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TNF P01375 4/20 0.42
EGFR P00533 1/20 0.32
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18151470 1.00 TNF (0.42) TNFEGFRMTOR
SCHEMBL18150889 0.87 TNF (0.47) TNFMTOR
SCHEMBL18151394 0.87 TNF (0.47) TNFMTOR
SCHEMBL18151826 0.85 EGFR (0.35) TNFEGFRMTOR
SCHEMBL18150789 0.85 TNF (0.43) TNFMTOR
SCHEMBL18151222 0.83 TNF (0.44) TNFMTOR
SCHEMBL29795004 0.83 TNF (0.44) TNFMTOR
SCHEMBL29795029 0.83 TNF (0.45) TNFMTOR
SCHEMBL18150324 0.83 TNF (0.45) TNFMTOR
SCHEMBL18151698 0.80 NTRK1 (0.41) TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4493221-A2 TARGETED BIFUNCTIONAL DEGRADERS Yale University (US) 2025-01-22 EP disclosed
CN-119212727-A Targeted bifunctional degradants 耶鲁大学 2024-12-27 CN disclosed
WO-2024182772-A2 MANNOSE 6-PHOSPHATE RECEPTOR BINDING COMPOUNDS FOR THE DEGRADATION OF EXTRACELLULAR PROTEINS AVILAR THERAPEUTICS, INC. (US) 2024-09-06 WO disclosed
WO-2023178199-A2 TARGETED BIFUNCTIONAL DEGRADERS YALE UNIVERSITY (US) 2023-09-21 WO disclosed
EP-4041262-A1 TARGETED BIFUNCTIONAL DEGRADERS Yale University (US) 2022-08-17 EP disclosed